Allergic reactions in children cause concern for parents. To relieve unpleasant symptoms and help the baby, antiallergic and antihistamines are prescribed. They have a quick effect on the body, relieve itching and redness.
Fenistil drops for children are an antihistamine and antiallergic drug. The dosage form is convenient for treatment. The product is safe for children from 1 month of age, has a minimum list side effects.
The drug relieves allergies, relieves serious conditions with various pathologies. Active ingredients block the production of histamine, so itching and redness of the skin disappears, puffiness is eliminated.
When Fenistil drops are prescribed for children:
Fenistil drops are often prescribed 3 days before vaccinations in order to reduce the effect of drugs on the baby's body. You need to know that the remedy does not cure, but only relieves the symptoms of allergies.
It is quite convenient to take drops for children. They can be added to water or breast milk for babies, or used undiluted for teens and adults.
Drops are available in small dark glass bottles of 20 ml. The cap is equipped with a built-in dosing dropper, which makes it easy to give the drug to the baby. The kit includes instructions in Russian.
Composition for 1 ml of the preparation:
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The liquid is transparent, odorless. It is allowed to use the drug for children under one year old.
Properties medicinal product are based on blocking histamine H1 receptors. Fenistil effectively fights itching and allergies. It has a mild sedative effect, as it affects the central nervous system.
The drops are stored in a dark and cool place, away from children. Shelf life from the date of opening is 2 years. In pharmacies, the drug is sold without a prescription.
Fenistil relieves itching, redness, has a mild anesthetic effect. It is absorbed by the body almost completely, it penetrates well into the tissues.
Indications for admission are:
You can take drops only as directed by your doctor. For children under one year old, the drug should not be abused, since there is a high likelihood of problems with the respiratory system.
Contraindications:
Fenistil rarely causes side effects. But in some cases, the patient's condition may worsen.
In the first trimester, taking the drug is completely prohibited. In the second and third, the treatment is carried out under the supervision of a physician.
Side effects of drops:
Drops are taken orally. The dosage and time of treatment are determined by the doctor, based on the diagnosis and the patient's age.
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For newborn babies, drops are added immediately before feeding in a bottle with a warm breast milk or a mixture. The product has a pleasant taste, which allows you to give it undiluted with a spoon.
For premature babies, the medicine is dosed based on the weight of the baby. First, the daily rate is calculated, then it is divided into 3 equal doses. It is allowed, in order to reduce drowsiness in children, to give a dose of a smaller volume in the morning, and a larger one in the evening.
The treatment period lasts 7-10 days. For chronic allergies, the drug is given in courses, with breaks of 5 days. Long-term use of the drug should be avoided.
How to use:
To prepare for vaccination, Fenistil is given within 3 days before vaccinations and 1-2 days after. This avoids drug-induced allergies.
Fenistil is a rather expensive drug, its average cost is 600 rubles. There are cheaper analogs with similar properties. Before replacing a prescribed drug with another, you should consult with your doctor.
Fenistil drops, intended for oral administration, are an anti-allergy agent.
Tradename: Fenistil®
Formula: 2- (2-dimethylaminoethyl) -3 - (1H) -indene maleate
Description: The drug is a clear liquid, colorless and odorless.
The drug is poured into 20 milliliters in tinted glass vials, which are equipped with a polypropylene cap, which, in turn, is equipped with a system that controls the first opening. Each bottle has a dropper dispenser and, accompanied by instructions for use, is packed in an individual cardboard box.
The active substance of Fenistil drops is dimethindene maleate. One milliliter of the finished preparation contains one milligram of it, supplemented with inactive substances: non-crystallized liquid sorbitol, sodium dihydrogen phosphate dihydrate, methyl parahydroxybenzoate, 96% ethanol and purified water.
The vial with the drug should be stored placed in its cardboard packaging in a place that is inaccessible to children. The room temperature should not exceed 30 degrees.
The use of the drug is possible within three years from the date of manufacture. It is not recommended to use it after the expiration date.
The drug Fenistil is an antihistamine, antiallergic, and antipruritic agent. As a blocker of H1-histamine receptors, it acts as a competitive histamine antagonist.
By its effect, the drug is able to reduce the increased capillary permeability, which is associated with an allergic reaction.
Drops can also have antikininic and not strong anticholinergic effects. With a daily intake of the drug, a slight sedative effect is possible.
The use of the drug Fenistil is indicated for the following ailments:
Taking the drug Fenistil is contraindicated for taking if the patient has signs of hypersensitivity to the components of the drug, especially to its active substance.
Also, drops should not be prescribed for angle-closure glaucoma, prostatic hyperplasia, as well as for infants under one month of age. The drug for premature babies is strongly not recommended for use.
The drug Fenistil is intended for internal use.
20 drops of the drug contain 1 milligram of the active substance.
These tables contain the dosage for children for three times a day.
Adult patients and adolescents who have reached the age of twelve daily dose can be prescribed in the amount of 3 to 6 milligrams (60-120 drops), which is divided into three doses of 20-40 drops three times a day.
Those patients who are prone to drowsiness can be prescribed as follows: 40 drops at night and 20 drops in the morning at breakfast.
For women during lactation, the drug is prescribed with caution.
To use Fenistil during pregnancy is allowed only when the benefits that are expected for the expectant mother may exceed the potential threat to the child. It is possible to use the drug only under the supervision of a doctor.
The drug Fenistil is prohibited to prescribe to newborn children.
Also, drops are prescribed with caution for children under one year old, since the manifestation of a sedative effect in such babies can be accompanied by sleep disturbances with periodic cessation of breathing.
Symptoms of excessive intake of the drug in adults will be manifestations of drowsiness and depression of the central nervous system. Children, in case of an overdose, can be overly agitated.
Manifestations of tachycardia, hallucinations, tonic-clonic seizures, mydriasis, dry mouth may also occur, and blood may “rush” to the face, urinary retention and fever may occur; there is a state of decreasing blood pressure, collapse.
Treatment can be carried out with activated charcoal, saline laxatives, drugs that support the activity of the cardiac and respiratory systems, except for analeptic drugs.
The drug is able to exert on the body and a number of unwanted influences as:
With the simultaneous administration of a drop of Fenistil, they are capable of enhancing the action of anxiolytics, a hypnotic drug.
When used together with ethanol, you can get a noticeable slowdown in the rate of reactions.
Co-administration of the drug with tricyclic antidepressants and anticholinergic drugs can increase the risk of increased intraocular pressure.
MAO inhibitors are able to enhance anticholinergic and depressive actions of the central nervous system.
Analogs of FENISTIL are those drugs that are similar to it in indications and pharmacology. In order to compare them, you need to pay attention to the substance that plays the role of an active one in the composition of the drug. In more expensive analogs, as a rule, there is a content of additives that enhance the effect of the active substance of the drug.
It should be remembered: the decision that the drug Fenistil should be replaced by any of its analogs can only be made by a doctor.
The drug can be purchased at any pharmacy where it is dispensed without a doctor's prescription. The drug is quite expensive - its approximate cost is about three hundred rubles.
Young mothers often encounter allergic reactions of their children to food or medicine and wonder how to reduce or eliminate the manifestations of allergies in their baby's body.
Fenistil for children is a modern antihistamine that should be in every mother's medicine cabinet from the first days of the long-awaited baby's birth. Fenistil replaced the outdated Suprastin and Tavegil counterparts.
The main substance in Fenistil, an effective and fast acting antihistamine, is dimethindene maleate, which has a sedative and antipruritic effect. This substance narrows the capillaries and reduces the expression of allergies. Additional components of the drug depend on the type of release.
The drug has the following properties:
The action of "Fenistil" is as follows:
The medication enters the bloodstream and is excreted from the body with bile and urine.
Produced in the form of drops or capsules, the product is designed for internal use by children and adults, it is prescribed in the following cases:
It is especially worth noting that it is contraindicated to prescribe Fenistil for newborn children (from the moment of birth to one month).
It is forbidden to use:
If your baby has a fever, use or - these are popular and effective means with a minimum of side effects.
Produced for children in several forms:
Internal medicine in the form of tablets or drops acts instantly, maintaining its effect for twelve hours. If mom decided to give "Fenistil" as prophylactic before vaccination, then this must be done no more than twelve hours before vaccination.
Fenistil for babies is also available in drops. When calculating children's daily allowance for Fenistil drops, young mothers need to proceed from the calculation of 0.1 mg of active active substance per one kilogram of the child's weight. Twenty drops contain 1 mg of active ingredient.
Calculation example: a baby is 4 months old and weighs 5 kg. thus, the calculation of the daily dose looks like this.
0.1 mg (dimethindene) multiplied by the weight 5 (kg) = 0.5 mg (10 drops).
Since there are three doses per day, then we divide 10 drops by three and get 3 drops per dose.
To consume the drops, mix them with a warm, but not hot drink or food and divide the dose of the medicine into three portions for gradual intake.
If the symptoms have partially disappeared within a week of taking Fenistil, parents should consult a doctor.
Before and after vaccination
The doctor advises to use before vaccination this drug because it helps to reduce the reaction of vaccination to the body, but only a few days before it, and not to use the drug for a day or two before vaccination. As this can affect vaccination results and change results, misinterpretation will arise.
If mothers decide to give a medication before vaccinating a baby with DPT, then this must be done as follows:
This type of medicine is used since the birth of a child.
Application rules:
Tablets are given to children only after 12 years, one piece per day for a course of no more than twenty-five days.
Admission rules:
Side effects when taken are extremely rare.
Before taking the medicine, you should consult with a pediatrician who correctly diagnosed and prescribe the appropriate treatment and dosage.
It is strictly forbidden to prescribe "Fenistil" on your own or to increase its dosage without the recommendation of a specialist.
In case of an overdose, the deterioration of the child's condition is predictable:
In case of an overdose, it is necessary to give the baby activated charcoal and to maintain respiratory and heart function.
If there are signs of intolerance, it is necessary to stop taking and consult a pediatrician about replacing the drug with analogues:
Mothers should pay attention to the fact that Fenistil's analogues have a number of contraindications, therefore, before taking other medications, it is necessary to consult a doctor. For example, "Zyrtec" and "Zodak" are drugs of the second generation, and "Fenistil" is of the first generation, "Zyrtec" has a number of side effects, and "Zodak" is allowed for admission to children only over one year old.
Let's compare analogs with Fenistil:
It is necessary to store the medicine for three years from the date of release, in a dry, dark place, protected from children, preferably in a refrigerator. In pharmacies "Fenistil" is dispensed without a doctor's prescription.
Active substance: dimethindene maleate.
1 ml of drops contains 1 mg of dimethindene maleate
Excipients: disodium phosphate dodecahydrate, citric acid monohydrate, benzoic acid, disodium edetate, sodium saccharin, propylene glycol, purified water.
Antihistamine for systemic use. CodeATX: R06AB03
Pharmacological properties
Pharmacodynamics
Antihistamine, anti-allergic and antipruritic agent. H1-histamine receptor blocker, is competitive antagonist histamine.
The drug reduces the increased capillary permeability associated with allergic reactions.
It also has antikinin and weak anticholinergic effects. When taking the drug during the day, there may be a slight sedation.
Pharmacokinetics
Quickly and completely absorbed when taken orally. Bioavailability is about 70%. The onset of action can be expected in 30 minutes and the main effect within 5 hours. The time to reach the maximum concentration of dimethindene in the blood plasma after oral administration of drops is observed within 2 hours. The connection with plasma proteins is 90%. Penetrates well into tissues. It is metabolized in the liver by hydroxylation and methoxylation. The half-life is 6 hours. It is excreted in the bile and urine (90% as a metabolite and 10% unchanged).
Symptomatic treatment of allergic diseases: urticaria, allergic diseases of the upper respiratory tract such as hay fever and year-round allergic rhinitis, food and drug allergies.
Itching of various origins, with the exception of itching with cholestasis. Itching for conditions with a rash such as chicken pox... Itching after insect bites.
As an adjuvant for eczema and other itchy dermatoses of allergic origin.
Hypersensitivity to dimethindene and other components that make up the drug. Childhood up to 1 month, especially premature ones.
Caution should be exercised when using the drug in patients with glaucoma, urinary retention in the presence of prostatic hyperplasia, bronchial asthma, chronic obstructive pulmonary disease, epilepsy.
Also, caution is required when prescribing Fenistil® NEW drops to children under the age of 1 year, since their sedation may be accompanied by episodes of sleep apnea.
The drug should be used in children aged 1 month to 1 year only on the recommendation of a doctor and only in case of strict medical indications. The recommended dose should not be exceeded.
Drops Fenistil ® NEW are ineffective for itching associated with cholestasis.
Application during pregnancy and breastfeeding
The use of Fenistil® NEW during pregnancy is possible on the recommendation of a doctor, only if the expected benefit to the mother outweighs the potential risk to the fetus. The use of the drug during breastfeeding is not recommended.
For oral administration.
Children under 12 years old:
For children, the usual daily dose is approximately 0.1 mg / kg body weight, i.e. 2 drops / kg of body weight. The daily dose should be divided into 3 doses.
For children aged 1 month to 12 years, the doses are shown in the table. Frequency rate of application - 3 times a day.
Children under 1 year old can use drops only on the recommendation of a doctor.
20 drops = 1 ml = 1 mg of dimethindene maleate.
Children over 12 years old and adults:
For adults and children over 12 years of age, the daily dose is usually 3-6 mg (60-120 drops), divided into 3 doses, that is, 20-40 drops 3 times a day.
Special patient populations
There is no data confirming that a dose adjustment is required for elderly patients (over 65 years old), patients with impaired liver and kidney function.
Mode of application
The drops can be taken with or without food. If used in infants, they should be added to the warm baby food bottle just before feeding. Fenistil® NEW drops should not be exposed to high temperatures. If the baby is already spoon-fed, the drops can be given undiluted. The drops taste good.
If you miss a dose, take the medicine as soon as you remember the missed dose, but no later than 2 hours before your next dose. If there are less than 2 hours before your next dose, do not take the missed dose, but take the next dose according to your medication schedule. Do not take a double dose instead of a missed one.
Side action
The most common side effects are fatigue, drowsiness, and nervousness.
Such side effects as agitation, headache, dizziness, gastrointestinal upset, nausea, dry mouth and throat.
Very rarely, anaphylactic reactions may occur, including facial edema, laryngeal edema, rash, muscle cramps, and shortness of breath.
If the listed adverse reactions or reactions not listed in this leaflet, you should see your doctor.
Symptoms: depression of the central nervous system (CNS) and drowsiness (mainly at adults), stimulation of the central nervous system and anticholinergic effects (especially in children), incl. agitation, ataxia, tachycardia, hallucinations, tonic-clonic seizures, mydriasis, dry mouth, flushing of the face, urinary retention and fever; decline blood pressure, collapse. Treatment: activated charcoal, saline laxatives, medicines to support the activity of the cardiac and respiratory systems. Stimulants should not be used.
Interaction with other medicinal products
The simultaneous use of drugs that have a depressing effect on the central nervous system can cause an increase in their action. Do not use the drug simultaneously with opioid analgesics, anticonvulsants, antidepressants (tricyclic antidepressants and monoamine oxidase inhibitors), antiemetics, antipsychotics, anxiolytics, sleeping pills and alcohol, because this can enhance the CNS depressant effect.
One of the most popular anti-allergic products for children. The drug effectively eliminates puffiness and itching of the skin, due to which it is prescribed as symptomatic remedy with viral and dermatological diseases. It has a high safety profile, it can be prescribed even during the neonatal period.
One of the dosage forms of the drug are drops for oral administration, produced in 20 ml each in a dropper bottle.
Drops for oral administration are a colorless transparent liquid that is almost odorless.
1 ml, which corresponds to 20 drops, contains 1 mg of dimethindene maleate.
As auxiliary components in the composition dosage form includes:
The medication is available in dark glass vials, which are equipped with a dropper dispenser for convenience. The volume of the dosage form is 20 ml.
Dimethindene maleate is a histamine H 1 receptor blocker, a competitive histamine antagonist. It relieves allergies, eliminates itching, excessive capillary permeability, which is observed during an allergic reaction. It has an anti-bradykinin and a weak m-anticholinergic effect. When taking the medication during the day, a mild sedative effect may appear.
After oral administration, the antihistamine effect of the medication begins in half an hour and reaches its maximum severity within 5 hours.
After oral administration, the active substance is rapidly absorbed. The maximum concentration in the blood is observed after 2 hours. The bioavailability of the drug reaches 70%. Up to 90% of the active substance binds to proteins, migrates well into tissues. Passing through the liver, the drug is metabolized.
The half-life reaches 6 hours. The drug is excreted through the intestines and kidneys: 90% of the active substance is excreted in the form of metabolites, the rest is unchanged.
Fenistil drops are prescribed when:
In addition, drops are prescribed to prevent allergies during hyposensitizing therapy.
Fenistil drops are not prescribed if there is:
The drug is not prescribed for babies under 1 month old. The drug is not prescribed in the first trimester of pregnancy, starting from the 14th week of gestation, it can be prescribed when the benefit to the woman outweighs the risk to the fetus. Treatment with Fenistil drops is incompatible with breastfeeding, therefore, during lactation, it is advisable to transfer the child to a mixture.
With caution, the drug should be prescribed to persons suffering from chronic obstructive pulmonary pathologies, epilepsy, infants aged 1 to 12 months, since their sedative effect may be accompanied by sleep apnea syndrome.
Method of administration and dosage
Fenistil drops are taken orally. The dosage of the drug is selected individually, depending on the age and weight of the child.
While taking Fenistil drops, there may be such undesirable reactions as:
If there is an aggravation of the above-listed adverse reactions or the occurrence of new ones, then it is worth informing the pediatrician about this.
Fenistil enhances the effect of anxiolytics, hypnotics and other medicines that have a depressing effect on the nervous system, namely:
Tricyclic antidepressants and m-anticholinergics, including bronchodilators and antispasmodics, increase the likelihood of developing glaucoma or urinary retention.
Do not take Fenistil and Prokabazin drops in parallel.
In children under 6 years of age, while taking Fenistil drops, excessive excitability may be observed.
The drug should not be exposed to high temperatures. For infants, it can be added to a bottle of warm baby food and given right before feeding, or spooned undiluted. The medicine tastes good.
The medication does not relieve itching caused by cholestasis.
There is no specific antidote, the victim is given saline laxatives. In addition, he is prescribed activities to help maintain the efficiency of the cardiovascular and respiratory systems. The victim should not be prescribed analeptics.
Fenistil drops should be stored at a temperature of a maximum of 25 degrees, out of the reach of children, in their original packaging. The shelf life of the medicinal product is 24 months.
Despite the fact that Fenistil drops are non-prescription drugs, self-medication with them is unacceptable, since only a doctor can choose the correct therapy regimen.